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HR+ / HER2− Advanced Breast Cancer — Systemic Therapy
First-line
Second-line
Later-line
SECOND-LINE
THIRD-LINE / LATER
HR+ / HER2−
advanced breast
cancer
Endocrine-sensitive
ESR1 mutation
PIK3CA / AKT / PTEN
PIK3CA mutation
gBRCA1/2
Endocrine-resistant
ADC by HER2 status
Frontline
CDK4/6 inhibitor + ET
MONALEESA / PALOMA ↗
Oral SERD
Elacestrant
EMERALD ↗
AKT pathway
Capivasertib + fulvestrant
CAPItello-291 ↗
PI3K
Alpelisib + fulvestrant
SOLAR-1 ↗
PARP
Olaparib / talazoparib
OlympiAD ↗
PIK3CA
Palbo + fulvestrant + inavolisib
INAVO120 ↗
No driver
Everolimus + AI / fulvestrant
BOLERO-2 ↗
HER2-low
Trastuzumab deruxtecan
DESTINY-Breast04 ↗
TROP2
Datopotamab deruxtecan
TROPION-Breast01 ↗
TROP2
Sacituzumab govitecan
TROPiCS-02 ↗